Reise-Engletten: Full Drug Profile
Reise-Engletten - General Information
Reise-Engletten (Dramamine, Gravol and Vertirosan) is an over-the-counter drug used to prevent motion sickness. It is closely related to diphenhydramine HCl, or Benadryl. It is primarily a H1-antagonist, but also possesses an antimuscarinic effect.
Pharmacology of Reise-Engletten
Reise-Engletten is an antiemetics drug combination that contains diphenhydramine and theophylline. It is not effective in the treatment of nausea associated with cancer chemotherapy. Reise-Engletten directly inhibits the stimulation of certain nerves in the brain and inner ear to suppress nausea, vomiting, dizziness, and vertigo.
Reise-Engletten for patients
Reise-Engletten Interactions
Dimenhydrinate may decrease emetic response to apomorphine.
Reise-Engletten Contraindications
Dimenhydrinate may impede diagnosis of appendicitis and may obscure signs of overdose.
Additional information about Reise-Engletten
- Reise-Engletten Indication
Used for treating vertigo, motion sickness, and nausea associated with pregnancy.
- Mechanism Of Action
- The mechanism by which some antihistamines exert their antiemetic, anti–motion sickness, and antivertigo effects is not precisely known but may be related to their central anticholinergic actions. They diminish vestibular stimulation and depress labyrinthine function. An action on the medullary chemoreceptive trigger zone may also be involved in the antiemetic effect.
- Drug Interactions
- Donepezil Possible antagonism of action
- Food Interactions
- Avoid alcohol.
- Generic Name
- Dimenhydrinate
- Synonyms
- Diphenhydramine Theoclate; Diphenhydrinate
- Drug Category
- Antiemetics; Histamine H1 Antagonists
- Drug Type
- Small Molecule; Approved
- Other Brand Names containing Dimenhydrinate
- Amosyt; Anautine; Andramine; Antemin; Aviomarin; Chloranautine; Diamarin; Dimate; Dimenest; Dimentabs; Dramalen; Dramamin; Dramarin; Dramilin; Dramyl; Dromyl; Eldodram; Gravinol; Gravol; Hydrinate; Menhydrinate; Neo-Navigan; Novamine; Permital; Reise-Engletten; Supremal; Teodramin; Travelin; Travelmin; Troversin; Vomex A; Xamamina;
- Absorption
- Well absorbed after oral administration.
- Toxicity (Overdose)
- Symptoms of overdose include delerium and hallucinations.
- Protein Binding
- 98 to 99%.
- Biotransformation
- Hepatic (cytochrome P-450 system).
- Half Life
- 1 to 4 hours
- Dosage Forms of Reise-Engletten
- Solution Intravenous
- Chemical IUPAC Name
- 2-benzhydryloxyethyl-dimethylazanium; 8-chloro-1,3-dimethyl-2-oxopurin-6-olate
- Chemical Formula
- C24H28ClN5O3
- Dimenhydrinate on Wikipedia
- https://en.wikipedia.org/wiki/Dimenhydrinate
- Organisms Affected
- Humans and other mammals
