Neodin-Depositum: Full Drug Profile
Neodin-Depositum - General Information
Neodin-Depositum is a mineralocorticoid hormone and an analog of desoxycorticosterone. It is white, odorless, and stable in air. It is practically insoluble in water, sparingly soluble in acetone, slightly soluble in methanol, ether and vegetable oils. Federal (U.S.A.) law restricts this drug to use by or on the order of a licensed veterinarian.
Pharmacology of Neodin-Depositum
Used to treat adrenocortical insufficiency, desoxycorticosterone pivalate is a mineralocorticoid hormone and an analogue of desoxycorticosterone. It primarily acts on the metabolism of sodium, potassium and water. When the drug is given, there is decreased excretion of sodium accompanied by increased excretion of potassium; the concentration of sodium in the blood is thereby increased whereas that of potassium is decreased. There is a concomitant increase in the volume of blood and extracellular fluids, with a fall in hematocrit. It increases the rate of renal tubular absorption of sodium.
Neodin-Depositum for patients
Neodin-Depositum Interactions
Neodin-Depositum Contraindications
Desoxycorticosterone Pivalate is contraindicated in patients with systemic fungal infections and in those with a history of possible or known hypersensitivity to this agent.
Additional information about Neodin-Depositum
- Neodin-Depositum Indication
For treatment of adrenocortical insufficiency especially in multiple sclerosis, congenital cerebral palsy, polyarteritis nodosa, and rheumatoid arthritis.
- Mechanism Of Action
- Neodin-Depositum binds to the mineralocorticoid receptor. Mineralocorticoids are a family of steroids, secreted by the adrenal cortex, necessary for the regulation of a number of metabolic processes including electrolyte regulation. Desoxycorticosterone pivalate exerts its effect through its interaction with the mineralocorticoid receptor (MR), whereby it reacts with the receptor proteins to form a steroid-receptor complex. This complex moves into the nucleus, where it binds to chromatin which results in genetic transcription of cellular DNA to messenger RNA. The steroid hormones appear to induce transcription and synthesis of specific proteins, which produce the physiological effects seen after administration.
- Generic Name
- Desoxycorticosterone Pivalate
- Synonyms
- DOCP; Desoxycortone Pivalate; Desoxycorticosterone Trimethylacetate; Deoxycortone Trimethylacetate; Deoxycortone Pivalate; Deoxycortolone Pivalate; Deoxycorticosterone Trimethylacetate; Deoxycorticosterone Pivalate; DTMA
- Drug Category
- Diuretics; Anti-Addison Agents
- Drug Type
- Small Molecule; Approved
- Other Brand Names containing Desoxycorticosterone Pivalate
- Cortexone M; Neodin-Depositum; Percorten; Percorten M; Percorten Pivalate;
- Toxicity (Overdose)
- Symptoms of overdose include polyuria, polydipsia, increased blood volume, edema, and cardiac enlargement.
- Protein Binding
- 90%
- Chemical IUPAC Name
- [2-(10,13-dimethyl-3-oxo-1,2,6,7,8,9,11,12,14,15,16,17-dodecahydrocyclopenta[a]phenanthren-17-yl)-2-oxoethyl] 2,2-dimethylpropanoate
- Chemical Formula
- C26H38O4
- Organisms Affected
- Humans and other mammals
